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Product Description

PC-61-CP085 is a recombinant, Fc-engineered chimeric version of the original PC-61 (PC-61.5.3) antibody. The variable domain sequences are identical but the constant region sequences have been switched from rat IgG1, λ to mouse IgG2a, λ for optimal use in murine models. This Fc-engineered antibody is reported to deplete Treg cells within the blood, lymph nodes and tumor microenvironment, whereas the original hybrioma-derived rat antibody failed to show reduction of intratumoral Treg cells. The enhanced Treg depletion within the tumor microenvironment by the Fc-engineered antibody is attributed to increased engagement with activating murine Fc gamma receptors, overcoming resistance caused by intratumoral upregulation of the inhibitory receptor FcγRIIb. Additionally, species-matched chimeric antibodies exhibit regulated effector functions—including Fc receptor binding and complement activation—and result in less immunogenicity and formation of anti-drug antibodies (ADAs) than xenogenic antibodies in animal models. The highly controlled sequence and lack of genetic drift in recombinant antibodies provide more reliable and reproducible results over hybridoma derived antibodies.

The PC-61.5.3-CP085 monoclonal antibody reacts with mouse IL-2Rα also known as CD25, Ly-43, p55, or Tac. IL-2Rα is the 55 kDa ligand-binding subunit of the interleukin 2 receptor alpha chain. IL-2Rα expression is largely restricted to tumor-infiltrating Treg cells in mice. Alone, the IL-2Rα binds IL-2 with relatively low affinity however, when IL-2Rα associates with IL-2Rβ (CD122) and the common gamma chain (CD132) the complex binds IL-2 with high affinity. The PC-61.5.3 antibody has been shown to inhibit the binding of IL-2 to both the low and high affinity IL-2 receptor forms and block CD25‐dependent IL‐2 signaling.

References:
Arce Vargas, Frederick et al. “Fc-Optimized Anti-CD25 Depletes Tumor-Infiltrating Regulatory T Cells and Synergizes with PD-1 Blockade to Eradicate Established Tumors.” Immunity vol. 46,4 (2017): 577-586. doi:10.1016/j.immuni.2017.03.013

Huss, David J et al. “Anti-CD25 monoclonal antibody Fc variants differentially impact regulatory T cells and immune homeostasis.” Immunology vol. 148,3 (2016): 276-86. doi:10.1111/imm.12609

Solomon, Isabelle et al. “CD25-Treg-depleting antibodies preserving IL-2 signaling on effector T cells enhance effector activation and antitumor immunity.” Nature cancer vol. 1,12 (2020): 1153-1166. doi:10.1038/s43018-020-00133-0


Specifications

Isotype Mouse IgG2a
Recommended Isotype Control(s) RecombiMAb mouse IgG2a isotype control, anti-hen egg lysozyme
Recommended Dilution Buffer InVivoPure pH 7.0 Dilution Buffer
Immunogen IL-2-dependent cytolytic mouse T cell clone B6.1
Reported Applications Western Blot*
Flow Cytometry*
CD25‐dependent IL‐2 signaling blockade*
In-vivo regulatory T cell depletion*
Intratumoral Treg depletion*
*Reported for the original rat IgG1, λ antibody
Formulation PBS, pH 7.0
Contains no stabilizers or preservatives
Endotoxin ≤0.5EU/mg (≤0.0005EU/μg)
Determined by LAL assay
Purity ≥95%
Determined by SDS-PAGE
Sterility 0.2 µm filtration
Production Purified from mammalian cell supernatant in an animal-free facility
Purification Protein G
Molecular Weight 150 kDa
Murine Pathogen Tests Ectromelia/Mousepox Virus: Negative
Hantavirus: Negative
K Virus: Negative
Lactate Dehydrogenase-Elevating Virus: Negative
Lymphocytic Choriomeningitis virus: Negative
Mouse Adenovirus: Negative
Mouse Cytomegalovirus: Negative
Mouse Hepatitis Virus: Negative
Mouse Minute Virus: Negative
Mouse Norovirus: Negative
Mouse Parvovirus: Negative
Mouse Rotavirus: Negative
Mycoplasma Pulmonis: Negative
Pneumonia Virus of Mice: Negative
Polyoma Virus: Negative
Reovirus Screen: Negative
Sendai Virus: Negative
Theiler’s Murine Encephalomyelitis: Negative
Storage The antibody solution should be stored at the stock concentration at 4°C. Do not freeze.
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Additional Formats

  1. Catalog #CP084
    RecombiMAb anti-mouse CD25 (LALA-PG) Read more